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Montai

AI-enabled drug discovery that predictably unlocks hard to drug targets to transform chronic disease.

About Montai

Montai is a different kind of drug company, purpose-built to make big leaps forward in the predictable discovery of great drugs for chronic diseases.

Montai is pioneering at the intersection of machine learning, biology, and diverse untapped chemistry that is rich with potential solutions to disease — Anthromolecule™ compounds. Tested and refined through eons of human co-evolution through chronic consumption, the topologically rich structures across Anthromolecules offer opportunities to engage complex biological targets with precision and selectivity, making this diverse chemistry a privileged starting point for small molecule drugs.

What if AI could unlock the predictable discovery of transformative small molecule drugs for chronic disease?
What if AI could unlock the predictable discovery of transformative small molecule drugs for chronic disease?

Our Mission

Many of today's innovative therapies remain out of reach or insufficient for most patients. What's more, finding new oral medicines historically has been largely a trial-and-error endeavor with many of the most important validated biological pathways considered undruggable with small molecules. This is particularly true for inflammation and immune system disorders. Montai aims to change this.

  • 169M
    Adults living with
    inflammatory & immune diseases
  • 2/3
    Advanced therapies are injectable biologics
  • 97%
    Of patients Lack access to advanced therapies
  • 70-90%
    Prefer oral medicines over injectables

The CONECTA Platform

The CONECTA™ Platform is a new drug operating system enabling the predictable discovery of transformative small molecule drugs from our unique chemical space.

Diverse, Untapped Bioactive Chemical Space at Unprecedented Scale

Montai is aggregating and curating the world's largest, fully-annotated set of Anthromolecules - bioactive molecules humans have chronically consumed.

We have developed proprietary tools to generate and curate over 1 billion synthetically accessible analogs with good drug-like properties derived from Anthromolecules. This opens accessibility to this privileged diverse chemical space at scale for efficient drug development.

Embedded in this space are many proven molecular modalities for unlocking complex biology, such as covalent binders, allosteric inhibitors, molecular glues and protein-protein interaction inhibitors. Now we can search this space universally for the first time to find optimal solutions for complex biology.

Precision Pathway Connections to Target Biology

Powered by next-generation multimodal foundation models trained on billions of curated and proprietary data points, Montai's AI tools efficiently unlock precision connections between the diverse Anthromolecule chemical space and the known drivers of complex disease biology governing inflammation and immune diseases, creating new opportunities for pill-based medicines.

Integrated Decisioning

CONECTA supercharges drug discovery and development with incredible efficiency, insights, and capabilities. More and earlier integrative decision making across multiple differentiated candidates, plus candidate discovery from diverse chemotypes de-risks development and provides unprecedented optionality.

What would have taken 1,000 years of experimentation can be done in a day.

A graphic representation of Anthromolecules, highlighting the ratio of known versus FDA-approved.

Our Platform Visualized

Montai has built the world's leading AI to decode the language of Anthromolecule chemistry to predictably unearth and optimize nature's bioactive solutions.
See how we do it.

The CONECTA® pipeline

Montai is rapidly advancing a pipeline of small molecule programs against validated biological pathways in inflammation and immune diseases including many that have been undruggable until now.
Target Discovery Lead
Op.
IND
Enabling
Phase 1
NRF2 (MTAI-1025)
Ulcerative Colitis
FIH 2026
Transcription
Factor
Biologics
Replacement
Oncology Pfizer
  • 1B+
    Superior starting points for drug discovery
  • 12
    Pathways validated in CONECTA® platform
  • 4
    hard-to-drug targets drugged with new mechanisms

We envision a world where, instead of regular and costly infusions, a convenient and safe pill for long-term use effectively treats a chronic disease, where solutions exist for diseases that today have none.

We are climbing mountains with AI, determined to improve health outcomes for as many people as possible to reduce the growing and unsustainable burden of chronic disease.
Meet Our Team

Featured News

  • Montai Therapeutics Presents Preclinical Data on NRF2 Agonist in Ulcerative Colitis at ACAAI Annual Meeting

    Article
    Nov 6, 2025
    Read on Business Wire
  • Montai Therapeutics Appoints Hans Hull as Chief Operations Officer

    Article
    Oct 28, 2025
    Read on Business Wire
  • Montai Therapeutics Appoints Allison Bogosian, JD, as Chief People and Administrative Officer

    Article
    Apr 28, 2025
    Read on Business Wire
  • Spotlight: Montai Builds a Multimodal AI Platform for Drug Discovery Using NVIDIA NIM Microservices

    Article
    Sep 26, 2024
    Read on NVIDIA Technical Blog
  • Montai Therapeutics Appoints Renowned Chemical Innovator Larry Hamann to Company's Board of Directors, Convenes Multidisciplinary Scientific Advisory Board to Inform Strategic Momentum

    Article
    May 29, 2024
    Read on Business Wire
  • How 3 Mass. companies are using AI to design drugs

    Article
    Mar 19, 2024
    Read on WBUR
  • Breaking Boundaries in Chemical Combinatorics Machine Learning: Unveiling the ComboPath Model at NeurIPS 2023

    Article
    Dec 13, 2023
    Read on LinkedIn
  • Montai Health Appoints Christian Antoni, M.D., Ph.D., as Company's First Chief Medical Officer

    Press Release
    Oct 24, 2023
    Read on GlobeNewswire
  • Montai Health Adds Industry Leaders to its Board of Directors

    Press Release
    May 17, 2023
    Read on Business Wire
  • Flagship Pioneering Unveils Montai Health to Treat and Preempt Chronic Disease Afflicting Two Billion People Worldwide

    Press Release
    December 13, 2022
    Read on The PR Newswire

Join Us

We are growing our team of leaders, committed to finding breakthroughs to make a difference in as many lives as possible.
View Open Positions

Contact Us

  • Partnerships

    We welcome the opportunity to partner with experts across areas who share our passion for creating Anthromolecule™ medicines and want to collaborate to accelerate the development of safe, efficacious and accessible therapies across diseases.

    partnerships@montai.com
  • Press

    For media inquiries or the latest on research, thought leadership, company news, and events contact:

    press@montai.com